Ph.D. student, Department of Chemistry, University of Nizhny Novgorod
RESEARCH INTERESTS: DFT, molecular docking, colchicine, tubulin, antimitotic activity
EMAIL: maleev.alexandr@yandex.ru
AWARDS, INTERSHIPS AND GRANTS
1. The development of the hybrid materials fordrug delivery systems based on gold nanoparticles functionalized by the biomarkers (The Russian Foundation for Basic Research)
PUBLICATIONS
1. Ekaterina S. Shchegravina, Alexander A. Maleev, Stanislav K. Ignatov, Iuliia A. Gracheva, Andreas Stein, Hans-Günther Schmalz, Andrey E. Gavryushin, Anastasiya A. Zubareva, Elena V. Svirshchevskaya, Alexey Yu. Fedorov. Synthesis and biological evaluation of novel non-racemic indole-containing allocolchicinoids, European Journal of Medicinal Chemistry 141 (2017) 51–60 https://doi.org/10.1016/j.ejmech.2017.09.055
2. A.A. Maleev, A.Yu. Fedorov, S.K. Ignatov. Docking study of pirroloallocolchicinoids – colchicine-binding site ligands / 3rd Kazan Summer School on Chemoinformatics, 5–7 July 2017, Kazan / Book of Abstracts. – 2017. p. 57
3. A.A. Maleev, A.Yu. Fedorov, S.Yu. Bukhvalova, S.K. Ignatov. Antimitotical activity of novel functionalized colchicine analogues. A molecular docking study // 6-th School-Conference on Atomistic Simulation of Functional Materials (ASFM 2017) // 6-th School-Conference on Atomistic Simulation of Functional Materials (ASFM 2017 Winter), 7–8 December 2017, Moscow / Book of Abstracts. – 2017, p. 23.
4. A.A. Малеев, С.Ю. Бухвалова, А.Ю. Федоров, С.К. Игнатов. Оценка биологической активности функционализированных аналогов колхицина — потенциальных антимитотических агентов методом молекулярного докинга / Всероссийская конференция по квантовой и математической химии, 13–17 ноября, Уфа / Сборник тезисов. – 2017. c. 45